Category based on conventional use | Class | Subclass | Drugs |
Multipurpose analgesics | Glucocorticoids | – | Dexamethasone, prednisone, methylprednisone |
Antidepressants | Tricyclic | Amitriptyline, desipramine, nortriptyline | |
SNRIs | Duloxetine, minalcipran, desvenlafaxine | ||
SSRIs | Paroxetine, citalopram | ||
Other | Buproprion | ||
Alpha-2 adrenergic agonists | – | Tizanidine, clonidine | |
Cannabinoids | – | Dronabinol, nabilone, nabiximols | |
Topical analgesics | – | Local anesthetics, lidocaine, capsaicin, tricyclic antidepressants, NSAIDs, others | |
Botulinum toxin injections | – | – | |
Used for neuropathic pain | All multipurpose analgesics | Refer to above | Refer to above |
Antiseizure medications | – | Gabapentin, pregabalin, valproate, phenytoin, carbamazepine, oxcarbazepine, topiramate, lamotrigine | |
Sodium channel blockers | Sodium channel modulator | Lacosamide | |
Sodium channel blocker | Mexiletine, intravenous lidocaine | ||
NMDA receptor antagonists | – | Ketamine, memantine, dextromethorphan, amantadine | |
GABA agonists | GABAa agonists | Clonazepam | |
GABAb agonists | Baclofen | ||
Used for bone pain | Osteoclast inhibitors | Bisphosphonates | Pamidronate, zolendronate, ibandronate |
– | Calcitonin | ||
RANKL inhibitor | Denosumab | ||
Radiopharmaceuticals | – | Strontium-89, samarium-153, radium-223 | |
NSAIDs, glucocorticoids | – | – | |
Used for bowel obstruction | Anticholinergic drugs | – | Scopolamine, atropine, glycopyrrolate |
Somatostatin analog | – | Octreotide | |
Glucocorticoids | – | – |
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