Traditional* | IUPHAR* | Clinical Effects |
µ1 | MOP | Supraspinal analgesia |
Peripheral analgesia | ||
Sedation | ||
Euphoria | ||
Prolactin release | ||
µ2 | Spinal analgesia | |
Respiratory depression | ||
Physical dependence | ||
Gastrointestinal dysmotility | ||
Pruritus | ||
Bradycardia | ||
Growth hormone release | ||
κ1 | KOP | Spinal analgesia |
Miosis | ||
Diuresis | ||
κ2 | Psychotomimesis | |
Dysphoria | ||
κ3 | Supraspinal analgesia | |
δ | DOP | Spinal and supraspinal analgesia |
Modulations of µ-receptor function | ||
Nociceptin/orphanin | NOP | Anxiolysis |
Analgesia |
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